Head to head

Semaglutide vs Tirzepatide

These are the two most-searched compounds in the whole category, and they're genuinely close cousins — both weekly, both injectable, both titrated slowly upward. The questions people actually have are about how they differ mechanistically and what that means for tracking, not which is 'best' (that's a clinician's call).

The short answer. Both are once-weekly injectable incretin drugs for type-2 diabetes and weight management. The core difference is receptor coverage: semaglutide is a single GLP-1 receptor agonist, while tirzepatide is a dual GIP/GLP-1 agonist. Their half-lives are similar (about a week), so both titrate over months and both reward a written dose history.

Side by side

 SemaglutideTirzepatide
ClassGLP-1 & incretinsGLP-1 & incretins
FormInjectionInjection
Half-life≈ 7 days (168 h)≈ 5 days (120 h)
Storage
Dose unitsmg, mcg, mlmg, ml
FDA statusApprovedApproved

Facts from the Stack compound library. See the full pages: Semaglutide · Tirzepatide.

How they differ

Receptor targets

Semaglutide acts on the GLP-1 receptor alone. Tirzepatide is a dual agonist — it activates both the GIP and GLP-1 receptors. That added GIP activity is the headline pharmacological distinction between them.

Titration ladders

Both climb through defined steps over months. Semaglutide's common ladder is 0.25 → 0.5 → 1 → 1.7 → 2.4 mg; tirzepatide's is 2.5 → 5 → 7.5 → 10 → 12.5 → 15 mg. Because the numbers aren't interchangeable, a log that records the dose at each step is the only reliable history.

Half-life & cadence

Both sit around a one-week half-life, so both are once-weekly and both take roughly a month to approach steady levels. A missed week halves the level rather than zeroing it — which is exactly the kind of thing an 'in your system' curve makes visible.

Brand context

Each molecule is marketed under multiple brand names for diabetes and for weight management. We never use brand names in the library — the molecule is what matters for tracking, and brands are trademarks.

Tracking either one

Whichever you log, the workflow is the same in Stack: add it once, set the schedule, and let the app handle reminders, supply projection and an "in your system" curve from the half-life. Run both? Group them into one protocol you can pause together.

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Not medical advice. This page compares publicly-documented properties of two compounds for educational purposes. It does not recommend either one, or any dose. How we source →

Last reviewed 2026-06-11